SCHEMBL28512652

SCHEMBL28512652

O=C(NCC1CCN(Cc2ccc(F)c(F)c2)CC1)c1cncc(NC(=O)c2ccnc(NC(=O)C3CC3)c2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 19/20 1.00
ACHE P22303 16/20 1.00
BCHE P06276 1/20 0.65
MAPT P10636 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28905775 0.92 GSK3B (1.00) GSK3BACHEBCHEMAPT
SCHEMBL28906880 0.90 GSK3B (1.00) GSK3BACHEBCHE
SCHEMBL28505211 0.88 GSK3B (1.00) GSK3BACHEBCHEMAPT
SCHEMBL28905792 0.87 GSK3B (1.00) GSK3BACHEBCHEMAPT
SCHEMBL28517234 0.85 GSK3B (1.00) GSK3BACHEBCHE
SCHEMBL28906889 0.83 GSK3B (1.00) GSK3BACHEBCHEMAPT
SCHEMBL28510938 0.79 GSK3B (0.69) GSK3BACHEBCHEMAPT
SCHEMBL29960639 0.79 GSK3B (1.00) GSK3BACHEBCHEMAPT
SCHEMBL28906878 0.79 GSK3B (1.00) GSK3BACHEBCHEMAPT
SCHEMBL29960710 0.79 GSK3B (0.69) GSK3BACHEBCHEMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112047928-B Isonicotinamide AChE-GSK3 double inhibitor and preparation method and application thereof 中国药科大学 2022-09-23 CN claimed
CN-112047928-A Isonicotinamide AChE-GSK3 double inhibitor and preparation method and application thereof 中国药科大学 2020-12-08 CN claimed
CN-112047928-B Isonicotinamide AChE-GSK3 double inhibitor and preparation method and application thereof 中国药科大学 2022-09-23 CN disclosed
CN-112047928-A Isonicotinamide AChE-GSK3 double inhibitor and preparation method and application thereof 中国药科大学 2020-12-08 CN disclosed