SCHEMBL28513014

SCHEMBL28513014

C[C@@H](C(=O)O)c1ccc(-c2ccnc3ccc(F)cc23)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 7/20 0.51
AKR1C2 P52895 7/20 0.51
CYP2C19 P33261 3/20 0.45
CYP2C9 P11712 2/20 0.45
APP P05067 2/20 0.45
CYP3A4 P08684 1/20 0.45
IDO1 P14902 1/20 0.45
PTGS1 P23219 3/20 0.45
PTGS2 P35354 3/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
FABP2 P12104 1/20 0.45
TSHR P16473 1/20 0.45
AKR1C4 P17516 1/20 0.45
ADRA2B P18089 1/20 0.45
CHRM3 P20309 1/20 0.45
HTR2C P28335 1/20 0.45
DRD3 P35462 1/20 0.45
AKR1C1 Q04828 1/20 0.45
SLC22A6 Q4U2R8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28513016 1.00 AKR1C3 (0.51) AKR1C3AKR1C2CYP2C19CYP2C9APP
SCHEMBL28514483 0.84 IDO1 (0.45) AKR1C3AKR1C2IDO1AKR1C4AKR1C1
SCHEMBL28514481 0.84 IDO1 (0.45) AKR1C3AKR1C2IDO1AKR1C4AKR1C1
SCHEMBL28516866 0.82 IDO1 (0.42) AKR1C3AKR1C2IDO1AAK1SLC22A12
SCHEMBL28516867 0.82 IDO1 (0.42) AKR1C3AKR1C2IDO1AAK1SLC22A12
SCHEMBL28513610 0.81 IDO1 (0.56) CYP2C9CYP3A4IDO1PSEN1PSEN2
SCHEMBL28513612 0.81 IDO1 (0.56) CYP2C9CYP3A4IDO1PSEN1PSEN2
SCHEMBL28513031 0.78 PIK3CA (0.39) AKR1C3AKR1C2IDO1AAK1SLC22A12
SCHEMBL28513028 0.78 PIK3CA (0.39) AKR1C3AKR1C2IDO1AAK1SLC22A12
SCHEMBL25523411 0.73 AAK1 (0.44) IDO1AAK1PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110218182-B IDO inhibitors 南京亘泰医药技术有限公司 2021-01-26 CN disclosed