SCHEMBL28513612

SCHEMBL28513612

CC(C(=O)Nc1ccc(Cl)cc1)c1ccc(-c2ccnc3ccc(F)cc23)cc1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 16/20 0.56
TDO2 P48775 7/20 0.56
CYP2C9 P11712 4/20 0.56
CYP2C8 P10632 3/20 0.56
CYP3A4 P08684 1/20 0.56
KCNH2 Q12809 1/20 0.56
PSEN1 P49768 1/20 0.45
PSEN2 P49810 1/20 0.45
APH1B Q8WW43 1/20 0.45
NCSTN Q92542 1/20 0.45
APH1A Q96BI3 1/20 0.45
PSENEN Q9NZ42 1/20 0.45
AAK1 Q2M2I8 1/20 0.44
FFAR2 O15552 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28513610 1.00 IDO1 (0.56) IDO1TDO2CYP2C9CYP2C8CYP3A4
SCHEMBL28521383 0.87 IDO1 (0.53) IDO1TDO2CYP2C9CYP2C8CYP3A4
SCHEMBL28521384 0.87 IDO1 (0.53) IDO1TDO2CYP2C9CYP2C8CYP3A4
SCHEMBL28516326 0.82 IDO1 (0.47) IDO1TDO2CYP2C9CYP2C8CYP3A4
SCHEMBL28516327 0.82 IDO1 (0.47) IDO1TDO2CYP2C9CYP2C8CYP3A4
SCHEMBL28513016 0.81 AKR1C3 (0.51) IDO1CYP2C9CYP3A4PSEN1PSEN2
SCHEMBL28513014 0.81 AKR1C3 (0.51) IDO1CYP2C9CYP3A4PSEN1PSEN2
SCHEMBL28523040 0.80 IDO1 (0.47) IDO1TDO2CYP2C9CYP2C8CYP3A4
SCHEMBL28523042 0.80 IDO1 (0.47) IDO1TDO2CYP2C9CYP2C8CYP3A4
SCHEMBL28513119 0.79 CIT (0.54) IDO1TDO2CYP2C9CYP2C8CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110218182-B IDO inhibitors 南京亘泰医药技术有限公司 2021-01-26 CN disclosed