SCHEMBL28513666

SCHEMBL28513666

Cc1cc(I)nn1Cc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.47
RIPK1 Q13546 1/20 0.45
PTGS2 P35354 1/20 0.44
GAA P10253 3/20 0.44
POLB P06746 2/20 0.44
LMNA P02545 2/20 0.44
TSHR P16473 1/20 0.44
ALDH1A1 P00352 1/20 0.44
CASP3 P42574 1/20 0.44
NR1H3 Q13133 1/20 0.44
SENP8 Q96LD8 1/20 0.44
SENP7 Q9BQF6 1/20 0.44
SENP6 Q9GZR1 1/20 0.44
GRN P28799 1/20 0.43
SORT1 Q99523 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.42
HTR2A P28223 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3322508 0.81 LMNA (0.61) KDM4EPTGS2GAAPOLBLMNA
SCHEMBL18096004 0.80 KDM4E (0.51) KDM4EGAALMNAALDH1A1MEN1
SCHEMBL25212702 0.79 KDM4E (0.47) KDM4EPTGS2GAAPOLBLMNA
SCHEMBL19531685 0.79 KDM4E (0.47) KDM4EPTGS2GAAPOLBLMNA
SCHEMBL12062174 0.79 KDM4E (0.47) KDM4EPTGS2GAAPOLBLMNA
SCHEMBL17627070 0.79 KDM4E (0.56) KDM4EPTGS2GAAPOLBLMNA
SCHEMBL4092108 0.78 PTGER1 (0.70)
SCHEMBL28109720 0.77 SMN1; SMN2 (0.66) GAAPOLBLMNAALDH1A1CASP3
SCHEMBL14924173 0.77 GRN (0.49) KDM4EPTGS2GAAPOLBLMNA
SCHEMBL12050569 0.76 GRN (0.64) KDM4EGAAPOLBTSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117263942-A SHP2 phosphatase inhibitors and methods of use thereof 传达治疗有限公司 2023-12-22 CN disclosed
CN-112166110-B SHP2 phosphatase inhibitors and methods of use thereof 传达治疗有限公司 2023-08-11 CN disclosed
CN-112166110-A SHP2 phosphatase inhibitors and methods of use thereof 传达治疗有限公司 2021-01-01 CN disclosed