SCHEMBL28514735

SCHEMBL28514735

CCOS(=O)(=O)c1ccc(C)cc1OCc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 4/20 0.45
CYP19A1 P11511 3/20 0.43
MAPT P10636 2/20 0.43
MAPK1 P28482 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
PTGER1 P34995 2/20 0.42
PTGER4 P35408 2/20 0.42
PTGER3 P43115 2/20 0.42
PTGER2 P43116 2/20 0.42
MAOB P27338 1/20 0.41
LMNA P02545 3/20 0.41
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
KEAP1 Q14145 1/20 0.40
NFE2L2 Q16236 1/20 0.40
AR P10275 1/20 0.40
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29198633 0.90 MRGPRX4 (0.44) MRGPRX4CYP19A1MAPTMAPK1TDP1
SCHEMBL21647406 0.89 KDM4E (0.40) MRGPRX4CYP19A1MAPTMAPK1TDP1
SCHEMBL21647514 0.88 KDM4E (0.41) MRGPRX4MAPTMAPK1TDP1L3MBTL1
SCHEMBL21647535 0.88 KDM4E (0.41) MRGPRX4MAPTMAPK1TDP1L3MBTL1
SCHEMBL25360195 0.88 KDM4E (0.41) MRGPRX4MAPTMAPK1TDP1L3MBTL1
SCHEMBL28541204 0.87 MRGPRX4 (0.45) MRGPRX4MAOB
SCHEMBL29285393 0.86 KEAP1 (0.43) CYP19A1MAPTTDP1L3MBTL1MAOB
SCHEMBL10511076 0.85 MRGPRX4 (0.46) MRGPRX4CYP19A1MAPTMAPK1TDP1
SCHEMBL8369436 0.84 MAPT (0.49) MRGPRX4CYP19A1MAPTMAPK1TDP1
SCHEMBL21815478 0.84 MEN1 (0.47) MAPTMAPK1L3MBTL1LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115038704-A Nitrogen oxide donating PDE-5 and/or PDE-6 inhibitor compounds 日东制药股份有限公司 2022-09-09 CN disclosed
CN-112261970-A 3- (5-hydroxy-1-oxoisoindolin-2-yl) piperidine-2, 6-dione derivatives and their use in the treatment of IKAROS family Zinc finger 2(IKZF2) dependent diseases 诺华股份有限公司 2021-01-22 CN disclosed
CN-112218859-A Modulators of proteolysis and related methods of use 阿尔维纳斯运营股份有限公司 2021-01-12 CN disclosed