SCHEMBL28514741

SCHEMBL28514741

Cc1cccc(C#C/C(=N/O)c2ccccc2)c1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 4/20 0.41
VCP P55072 1/20 0.41
FFAR1 O14842 4/20 0.40
SMN1; SMN2 Q16637 1/20 0.38
S1PR2 O95136 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HSP90AA1 P07900 1/20 0.38
MAPT P10636 1/20 0.38
OPRK1 P41145 1/20 0.38
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
FFAR4 Q5NUL3 1/20 0.37
POLB P06746 1/20 0.36
CNR2 P34972 2/20 0.36
CNR1 P21554 1/20 0.36
PARP1 P09874 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28649093 1.00 GRM5 (0.41) GRM5VCPFFAR1SMN1; SMN2S1PR2
SCHEMBL28509399 0.91 VCP (0.44) GRM5VCPFFAR1SMN1; SMN2ALDH1A1
SCHEMBL28501871 0.83 APP (0.44) VCPSMN1; SMN2S1PR2ALDH1A1HSP90AA1
SCHEMBL28499562 0.82 VCP (0.60) VCPSMN1; SMN2ALDH1A1HSP90AA1MAPT
SCHEMBL28644592 0.82 VCP (0.51) GRM5VCPFFAR1SMN1; SMN2ALDH1A1
SCHEMBL28501872 0.82 VCP (0.51) GRM5VCPFFAR1SMN1; SMN2ALDH1A1
SCHEMBL31614569 0.78 VCP (0.68) GRM5VCPFFAR1SMN1; SMN2S1PR2
SCHEMBL5592873 0.78 VCP (0.68) GRM5VCPFFAR1SMN1; SMN2S1PR2
SCHEMBL141877 0.76 GRM5 (0.45) GRM5FFAR1FFAR4
SCHEMBL141876 0.76 GRM5 (0.45) GRM5FFAR1FFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112062735-B Synthesis method of isoselenazole derivative 温州大学 2022-11-08 CN disclosed
CN-112159364-B Synthetic method of isothiazole derivative 温州大学 2022-06-24 CN disclosed
CN-112159364-A Synthetic method of isothiazole derivative 温州大学 2021-01-01 CN disclosed
CN-112062735-A Synthesis method of isoselenazole derivative 温州大学 2020-12-11 CN disclosed