SCHEMBL28515978

SCHEMBL28515978

COc1cc(C=NNC(=O)c2ccc(O)c(OC)c2)ccc1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GAA P10253 6/20 0.81
KDM4E B2RXH2 2/20 0.81
GCGR P47871 4/20 0.78
MPO P05164 1/20 0.77
NT5E P21589 1/20 0.77
CA12 O43570 1/20 0.76
CA1 P00915 1/20 0.76
CA2 P00918 1/20 0.76
CA9 Q16790 1/20 0.76
KMT2A Q03164 5/20 0.76
MEN1 O00255 4/20 0.76
POLB P06746 6/20 0.75
MAPT P10636 2/20 0.73
ALDH1A1 P00352 1/20 0.73
PKM P14618 1/20 0.71
NR1I2 O75469 1/20 0.70
AHR P35869 1/20 0.70
SMN1; SMN2 Q16637 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28521274 0.95 GAA (0.77) GAAKDM4EGCGRMPONT5E
SCHEMBL28515502 0.92 GAA (0.81) GAAKDM4EGCGRMPONT5E
SCHEMBL28521660 0.92 GCGR (0.78) GAAKDM4EGCGRMPONT5E
SCHEMBL18642551 0.91 GAA (0.80) GAAKDM4EGCGRMPONT5E
SCHEMBL18642552 0.91 GAA (0.80) GAAKDM4EGCGRMPONT5E
SCHEMBL2542993 0.91 GAA (0.80) GAAKDM4EGCGRMPONT5E
SCHEMBL28520360 0.90 GAA (0.77) GAAKDM4EGCGRMPONT5E
SCHEMBL28521911 0.90 GAA (0.77) GAAKDM4EGCGRMPONT5E
SCHEMBL11157751 0.90 GAA (1.00) GAAKDM4EGCGRMPONT5E
SCHEMBL2663644 0.89 GCGR (0.74) GAAKDM4EGCGRKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112079744-B Aromatic acylhydrazone derivatives and application thereof as NA (adenosine) inhibitor 湖南大学 2021-07-30 CN claimed
CN-112079744-A Aromatic acylhydrazone derivatives and application thereof as NA (adenosine) inhibitor 湖南大学 2020-12-15 CN claimed
CN-112079744-B Aromatic acylhydrazone derivatives and application thereof as NA (adenosine) inhibitor 湖南大学 2021-07-30 CN disclosed
CN-112079744-A Aromatic acylhydrazone derivatives and application thereof as NA (adenosine) inhibitor 湖南大学 2020-12-15 CN disclosed