SCHEMBL28516401

SCHEMBL28516401

CONC(=O)c1ccc(N2CCN(C(=O)OC(C)(C)C)CC2)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.64
MAPT P10636 5/20 0.64
LMNA P02545 3/20 0.64
KMT2A Q03164 5/20 0.64
MEN1 O00255 3/20 0.64
CYP2C19 P33261 1/20 0.64
HTT P42858 2/20 0.62
NPSR1 Q6W5P4 1/20 0.62
ALDH1A1 P00352 3/20 0.58
GPR119 Q8TDV5 6/20 0.58
NAMPT P43490 1/20 0.54
TSHR P16473 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.50
ESR2 Q92731 1/20 0.48
NPC1 O15118 1/20 0.48
NR2F2 P24468 1/20 0.48
ESRRB O95718 1/20 0.48
ESR1 P03372 1/20 0.48
ESRRA P11474 1/20 0.48
ESRRG P62508 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20423694 0.88 KMT2A (0.68) SMN1; SMN2MAPTLMNAKMT2AMEN1
SCHEMBL2388387 0.85 MAPT (0.62) SMN1; SMN2MAPTLMNAKMT2AMEN1
SCHEMBL5573222 0.85 MAPT (0.76) SMN1; SMN2MAPTLMNAKMT2AMEN1
SCHEMBL29803251 0.85 MAPT (0.69) SMN1; SMN2MAPTLMNAKMT2AMEN1
SCHEMBL12720262 0.85 KMT2A (0.64) SMN1; SMN2MAPTLMNAKMT2AMEN1
SCHEMBL30182423 0.85 MAPT (0.69) SMN1; SMN2MAPTLMNAKMT2AMEN1
SCHEMBL13218466 0.84 GPR119 (0.79) SMN1; SMN2MAPTLMNAKMT2AMEN1
SCHEMBL1481563 0.82 GPR119 (0.78) SMN1; SMN2MAPTLMNAKMT2AMEN1
SCHEMBL63633 0.82 MAPT (0.65) SMN1; SMN2MAPTLMNAKMT2AMEN1
SCHEMBL24891935 0.82 MAPT (0.62) SMN1; SMN2MAPTLMNAKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110305062-B Substituted isoquinolone compound and synthesis method and application thereof 广州医科大学 2021-01-05 CN disclosed