SCHEMBL28517075

SCHEMBL28517075

O=C(O)c1cc2n(n1)CCCCC2

nearest known ligand 0.52

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.44
HTR2C P28335 1/20 0.44
LDHA P00338 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1423651 0.98 HTR2A (0.44) HTR2AHTR2CLDHA
SCHEMBL1423019 0.93 HTR2A (0.40) HTR2AHTR2CLDHA
SCHEMBL16794173 0.83 HTR2A (0.44) HTR2AHTR2CLDHA
SCHEMBL31389508 0.81 ALDH1A1 (0.42) HTR2AHTR2CLDHA
SCHEMBL25485602 0.79 HTR2A (0.44) HTR2AHTR2CLDHA
SCHEMBL18377472 0.79 POLB (0.46) HTR2AHTR2CLDHA
SCHEMBL22275219 0.79 ALDH1A1 (0.43) HTR2AHTR2CLDHA
SCHEMBL6379433 0.77 NPC1 (0.44) HTR2AHTR2C
SCHEMBL6381168 0.77 CYP1A2 (0.44)
Potassium Ion SCHEMBL5123542 0.76 HTR2A (0.39) HTR2AHTR2CLDHA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112204036-B Macrocyclic fused pyrazoles as MCL-1 inhibitors 苏州亚盛药业有限公司 2022-12-27 CN disclosed
CN-112204036-A Macrocyclic fused pyrazoles as MCL-1 inhibitors 苏州亚盛药业有限公司 2021-01-08 CN disclosed