SCHEMBL28517201

SCHEMBL28517201

O=[N+]([O-])c1ccc(Br)cc1OCCN1CCOCC1

nearest known ligand 0.70

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.61
CYP2D6 P10635 1/20 0.61
CYP2C19 P33261 1/20 0.61
ALDH1A1 P00352 7/20 0.57
MAPT P10636 2/20 0.57
HTT P42858 1/20 0.57
KDM4E B2RXH2 5/20 0.55
NPC1 O15118 2/20 0.55
RAB9A P51151 2/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
LMNA P02545 1/20 0.52
CHEK1 O14757 1/20 0.51
TP53 P04637 1/20 0.50
POLB P06746 2/20 0.49
TSHR P16473 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30104625 0.89 ALDH1A1 (0.64) ALDH1A1MAPTHTTKDM4ERAB9A
SCHEMBL20511532 0.89 ALDH1A1 (0.64) ALDH1A1MAPTHTTKDM4ERAB9A
SCHEMBL212946 0.85 CYP1A2 (0.65) CYP1A2CYP2D6CYP2C19ALDH1A1MAPT
SCHEMBL1926359 0.84 CYP1A2 (0.60) CYP1A2CYP2D6CYP2C19ALDH1A1MAPT
SCHEMBL1852361 0.82 CYP2D6 (0.88) CYP1A2CYP2D6CYP2C19ALDH1A1KDM4E
SCHEMBL1516573 0.82 ALDH1A1 (0.67) ALDH1A1MAPTHTTKDM4EMEN1
SCHEMBL17609969 0.80 CYP1A2 (0.57) CYP1A2CYP2D6CYP2C19ALDH1A1MAPT
SCHEMBL23628977 0.80 ALDH1A1 (0.58) CYP1A2CYP2D6CYP2C19ALDH1A1MAPT
SCHEMBL23325984 0.79 ALDH1A1 (0.56) CYP1A2CYP2D6CYP2C19ALDH1A1KDM4E
SCHEMBL14785100 0.79 ALDH1A1 (0.59) CYP1A2CYP2D6CYP2C19ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed