SCHEMBL28518062

SCHEMBL28518062

CC1(C(=O)Nc2nc3ccc(C(F)(F)F)cc3s2)CCCCCC1

nearest known ligand 0.65

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 2/20 0.65
CSNK1D P48730 13/20 0.61
ADORA1 P30542 2/20 0.59
CYP2D6 P10635 1/20 0.59
ACP1 P24666 1/20 0.56
LRRK2 Q5S007 1/20 0.52
ADORA2A P29274 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31236382 1.00 DYRK1A (0.65) DYRK1ACSNK1DADORA1CYP2D6ACP1
SCHEMBL28527314 1.00 DYRK1A (0.65) DYRK1ACSNK1DADORA1CYP2D6ACP1
SCHEMBL30944303 1.00 DYRK1A (0.65) DYRK1ACSNK1DADORA1CYP2D6ACP1
SCHEMBL28519830 0.99 DYRK1A (0.67) DYRK1ACSNK1DADORA1CYP2D6ACP1
SCHEMBL30944362 0.99 DYRK1A (0.67) DYRK1ACSNK1DADORA1CYP2D6ACP1
SCHEMBL30944395 0.84 DYRK1A (0.67) DYRK1ACSNK1DADORA1ACP1ADORA2A
SCHEMBL28522297 0.84 DYRK1A (0.67) DYRK1ACSNK1DADORA1ACP1ADORA2A
SCHEMBL28907246 0.84 DYRK1A (0.67) DYRK1ACSNK1DADORA1ACP1ADORA2A
SCHEMBL30944408 0.84 DYRK1A (0.67) DYRK1ACSNK1DADORA1ACP1ADORA2A
SCHEMBL30944285 0.83 DYRK1A (0.60) DYRK1ACSNK1DCYP2D6ACP1LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112423746-A Novel anti-mycobacterial heterocyclic amides 克莱斯通公司 2021-02-26 CN claimed
CN-112423746-A Novel anti-mycobacterial heterocyclic amides 克莱斯通公司 2021-02-26 CN disclosed