SCHEMBL28518271

SCHEMBL28518271

Fc1ccc(Oc2cc(Br)cc3[nH]cnc23)c(F)c1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 14/20 0.44
EPAS1 Q99814 1/20 0.38
MAP4K4 O95819 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
PRNP P04156 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
HTT P42858 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HSPB1 P04792 1/20 0.35
MAPK14 Q16539 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16738693 0.76 TRPA1 (0.46) TRPA1EPAS1MAP4K4MAPT
SCHEMBL1144726 0.72 MEN1 (0.44) MEN1ALDH1A1PRNPMAPTHPGD
SCHEMBL29804933 0.72 MEN1 (0.44) MEN1ALDH1A1PRNPMAPTHPGD
SCHEMBL22685864 0.71 BRD4 (0.43) MEN1ALDH1A1PRNPMAPTHPGD
SCHEMBL29745481 0.71 BRD4 (0.43) MEN1ALDH1A1PRNPMAPTHPGD
SCHEMBL10456772 0.70 TRPA1 (0.56) TRPA1EPAS1MAP4K4ALDH1A1HSPB1
SCHEMBL15403615 0.69 MAP4K4 (0.45) TRPA1EPAS1MAP4K4HTTKMT2A
SCHEMBL28509653 0.68 EPAS1 (0.43) TRPA1EPAS1MAP4K4ALDH1A1HSPB1
SCHEMBL30194212 0.68 EPAS1 (0.43) TRPA1EPAS1MAP4K4ALDH1A1HSPB1
SCHEMBL20160295 0.67 EPAS1 (0.44) TRPA1EPAS1ALDH1A1HPGDHSPB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112300154-B Nitrogen-containing heterocyclic compound, preparation method and application thereof 上海弘翊生物科技有限公司 2023-01-24 CN disclosed
CN-112300154-A Nitrogen-containing heterocyclic compound, preparation method and application thereof 上海弘翊生物科技有限公司 2021-02-02 CN disclosed