SCHEMBL28520050

SCHEMBL28520050

CCCC1(CCC)NC(=O)c2cc(N)ccc2O1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.34
RET P07949 5/20 0.33
ALK Q9UM73 2/20 0.33
FLT3 P36888 1/20 0.33
STK17B O94768 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
FTO Q9C0B1 1/20 0.32
RPS6KA3 P51812 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
ALDH1A1 P00352 2/20 0.30
NPC1 O15118 1/20 0.30
TP53 P04637 1/20 0.30
CYP3A4 P08684 1/20 0.30
TSHR P16473 1/20 0.30
MAPK1 P28482 1/20 0.30
RAB9A P51151 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29634186 1.00 CYP19A1 (0.34) CYP19A1RETALKFLT3STK17B
SCHEMBL29634370 0.88 NPSR1 (0.35) CYP19A1RETALKFLT3STK17B
SCHEMBL28524835 0.88 NPSR1 (0.35) CYP19A1RETALKFLT3STK17B
SCHEMBL28524406 0.79 CYP3A4 (0.46) MEN1KMT2AALDH1A1CYP3A4SMN1; SMN2
SCHEMBL29634252 0.79 CYP3A4 (0.46) MEN1KMT2AALDH1A1CYP3A4SMN1; SMN2
SCHEMBL28531506 0.77 RET (0.36) RETALKFLT3MEN1KMT2A
SCHEMBL29634201 0.77 RET (0.36) RETALKFLT3MEN1KMT2A
SCHEMBL7512827 0.71 ALDH1A1 (0.47) MEN1KMT2ANPSR1ALDH1A1NPC1
SCHEMBL29770999 0.71 ALDH1A1 (0.61) MEN1KMT2AFTORPS6KA3ALDH1A1
SCHEMBL28523381 0.70 ALDH1A1 (0.64) MEN1KMT2AFTOALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112442022-B Benzoxazine-4-ketone compound, preparation method and medical application thereof 承德医学院 2022-05-20 CN disclosed
CN-112442022-A Benzoxazine-4-ketone compound, preparation method and medical application thereof 承德医学院 2021-03-05 CN disclosed