SCHEMBL28520686

SCHEMBL28520686

NC(=O)C1(C(N)=O)CC1c1ccc(F)cc1F

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 3/20 0.43
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
HTR2B P41595 1/20 0.40
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
KDM1A O60341 2/20 0.38
KDM1B Q8NB78 1/20 0.38
KCNN4 O15554 4/20 0.37
PARP1 P09874 1/20 0.36
TP53 P04637 1/20 0.36
MC4R P32245 3/20 0.34
MC5R P33032 2/20 0.34
MC3R P41968 2/20 0.34
MC1R Q01726 2/20 0.34
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28521030 0.81 KDM1A (0.49) HTR2CHTR2BKDM1AKDM1BKCNN4
SCHEMBL2158810 0.80 OPRL1 (0.36) OPRL1
SCHEMBL5680300 0.79 MEN1 (0.39) OPRL1KDM1AKDM1B
SCHEMBL28520614 0.77 KDM1A (0.50) HTR2AHTR2CHTR2BCES2CES1
SCHEMBL2594172 0.76 KDM1A (0.44) HTR2CHTR2BKDM1AKDM1BKCNN4
SCHEMBL900614 0.76 KDM1A (0.45) KDM1AKCNN4KCNH2
Water SCHEMBL2458176 0.75 KDM1A (0.44) KDM1AKCNN4KCNH2
Hydrochloric Acid SCHEMBL29430083 0.75 KDM1A (0.47) KDM1AKCNN4KCNH2
SCHEMBL5899787 0.73 HTR2A (0.42) OPRL1HTR2AHTR2CHTR2BCES2
SCHEMBL28514962 0.72 HTR2A (0.38) HTR2AHTR2CHTR2BCES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112142619-B 1, 1-cyclopropane dicarboxylic acid amide compound and preparation method and application thereof 浙江工业大学 2023-01-10 CN disclosed
CN-112142619-A 1, 1-cyclopropane dicarboxylic acid amide compound and preparation method and application thereof 浙江工业大学 2020-12-29 CN disclosed