SCHEMBL5899787

SCHEMBL5899787

NCC1(C(=O)O)CC1c1ccc(F)cc1F

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
HTR2B P41595 1/20 0.42
OPRL1 P41146 2/20 0.38
KDM1A O60341 2/20 0.34
CES2 O00748 1/20 0.34
CES1 P23141 1/20 0.34
KDM1B Q8NB78 1/20 0.34
GRIN2B Q13224 2/20 0.34
LTB4R Q15722 1/20 0.34
LTB4R2 Q9NPC1 1/20 0.34
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
TP53 P04637 1/20 0.33
MC4R P32245 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5899779 0.89 KDM1A (0.44) KDM1ACES2CES1KDM1B
SCHEMBL5899780 0.82 KDM1A (0.47) HTR2AHTR2CHTR2BKDM1AKDM1B
SCHEMBL5899781 0.80 HTR2C (0.42) HTR2CHTR2BKDM1ACES2CES1
SCHEMBL5899774 0.80 KDM1A (0.49) HTR2AHTR2CHTR2BKDM1AGRIN2B
SCHEMBL5899615 0.79 KDM1A (0.44) HTR2AHTR2CHTR2BKDM1ASLC6A2
SCHEMBL5899701 0.78 HTR2C (0.38) HTR2CHTR2BKDM1ACES2CES1
SCHEMBL5899782 0.76 TUBB4A (0.32) KDM1ACES2CES1
SCHEMBL5899791 0.75 TRPA1 (0.40) HTR2AHTR2CGRIN2BLTB4RLTB4R2
SCHEMBL5899756 0.73 HTR2A (0.41) HTR2AHTR2CGRIN2B
SCHEMBL28520686 0.73 OPRL1 (0.43) HTR2AHTR2CHTR2BOPRL1KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7030267-B2 Cycloproply β-amino acid derivatives WARNER-LAMBERT COMPANY, LLC (US) 2006-04-18 US disclosed
US-20040147608-A1 Cyclopropyl beta-amino acid derivatives SCHWARZ JACOB BRADLEY (US) 2004-07-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040147608-A1 Cyclopropyl beta-amino acid derivatives CACNA1S, CACNA1D, CACNA1B HTR2A 235/4885HTR2C 285/4885HTR2B 392/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.