SCHEMBL28520979

SCHEMBL28520979

CC1CN(c2cccc3ccccc23)CCN1C(=O)OC(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.49
HDAC1 Q13547 1/20 0.47
GPR119 Q8TDV5 2/20 0.45
NR1H2 P55055 5/20 0.44
BACE1 P56817 1/20 0.43
NR1H3 Q13133 3/20 0.43
CYP11B2 P19099 1/20 0.43
SUV39H2 Q9H5I1 1/20 0.41
ACHE P22303 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17114986 0.87 MAP4K4 (0.47) MAP4K4HDAC1GPR119NR1H2CYP11B2
SCHEMBL17114988 0.87 MAP4K4 (0.47) MAP4K4HDAC1GPR119NR1H2CYP11B2
SCHEMBL30882769 0.86 NR1H2 (0.46) GPR119NR1H2BACE1NR1H3CYP11B2
SCHEMBL28584377 0.86 NR1H2 (0.46) GPR119NR1H2BACE1NR1H3CYP11B2
SCHEMBL25054057 0.86 NR1H2 (0.46) GPR119NR1H2BACE1NR1H3CYP11B2
SCHEMBL25054060 0.84 NR1H2 (0.59) NR1H2BACE1NR1H3CYP11B2ACHE
SCHEMBL30386832 0.84 NR1H2 (0.59) NR1H2BACE1NR1H3CYP11B2ACHE
SCHEMBL31082592 0.84 CYP11B2 (0.43) GPR119BACE1CYP11B2ACHE
SCHEMBL13999776 0.84 HDAC1 (0.49) MAP4K4HDAC1GPR119NR1H2NR1H3
SCHEMBL3621405 0.84 HDAC1 (0.52) MAP4K4HDAC1GPR119NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112341396-B Novel monoacylglycerol esterase inhibitor and preparation method and application thereof 四川大学华西医院 2022-07-26 CN disclosed
CN-112341396-A Novel monoacylglycerol esterase inhibitor and preparation method and application thereof 四川大学华西医院 2021-02-09 CN disclosed