SCHEMBL28522003

SCHEMBL28522003

CC(C)(C)OC(=O)NC1CCC(n2c(=O)[nH]c3ccccc32)CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.56
MAPK1 P28482 2/20 0.56
HSD11B1 P28845 4/20 0.52
TNKS O95271 3/20 0.51
PARP2 Q9UGN5 1/20 0.51
CHRM2 P08172 2/20 0.49
CHRM4 P08173 2/20 0.49
CHRM1 P11229 2/20 0.49
CHRM3 P20309 2/20 0.49
CHRM5 P08912 1/20 0.49
CCR5 P51681 1/20 0.49
OPRL1 P41146 1/20 0.47
KDM4E B2RXH2 1/20 0.47
PMP22 Q01453 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
TNKS2 Q9H2K2 1/20 0.47
OPRM1 P35372 2/20 0.47
OPRD1 P41143 1/20 0.47
OPRK1 P41145 1/20 0.47
OGFRL1 Q5TC84 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15289030 1.00 ALDH1A1 (0.56) ALDH1A1MAPK1HSD11B1TNKSPARP2
SCHEMBL22605771 1.00 ALDH1A1 (0.56) ALDH1A1MAPK1HSD11B1TNKSPARP2
SCHEMBL8863582 0.94 CHRM1 (0.59) ALDH1A1MAPK1HSD11B1CHRM2CHRM4
SCHEMBL8863635 0.94 CHRM1 (0.59) ALDH1A1MAPK1HSD11B1CHRM2CHRM4
SCHEMBL8863576 0.94 CHRM1 (0.59) ALDH1A1MAPK1HSD11B1CHRM2CHRM4
SCHEMBL22605489 0.91 ALDH1A1 (0.50) ALDH1A1MAPK1HSD11B1CHRM2CHRM4
SCHEMBL22588003 0.91 ALDH1A1 (0.50) ALDH1A1MAPK1HSD11B1CHRM2CHRM4
SCHEMBL30317025 0.91 ALDH1A1 (0.50) ALDH1A1MAPK1HSD11B1CHRM2CHRM4
SCHEMBL15289136 0.85 TNKS (0.46) ALDH1A1MAPK1TNKSPARP2TNKS2
SCHEMBL7184086 0.83 ALDH1A1 (0.49) ALDH1A1MAPK1HSD11B1TNKSPARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111848598-B Heterocyclic compound, application thereof and composition containing same 健艾仕生物医药有限公司 2024-12-10 CN disclosed
CN-111848598-A Heterocyclic ring-containing compound, application thereof and composition containing heterocyclic ring-containing compound 健艾仕生物医药有限公司 2020-10-30 CN disclosed