SCHEMBL28522151

SCHEMBL28522151

Fc1ccc2ccnc(F)c2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 5/20 0.42
MAPT P10636 2/20 0.41
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
CYP2A6 P11509 1/20 0.38
MAP3K14 Q99558 1/20 0.37
TYMS P04818 2/20 0.37
CCNC P24863 1/20 0.37
CDK8 P49336 1/20 0.37
CYP19A1 P11511 1/20 0.36
CDK2 P24941 2/20 0.36
CDC7 O00311 1/20 0.36
ROCK1 Q13464 1/20 0.36
CTDSP1 Q9GZU7 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
BACE1 P56817 1/20 0.35
PARP1 P09874 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12053800 0.79 TRPA1 (0.41) TRPA1MAPTCYP1A2CYP3A4CYP2D6
SCHEMBL17844959 0.79 TRPA1 (0.41) TRPA1MAPTCYP1A2CYP3A4CYP2D6
SCHEMBL1315422 0.79 MAPT (0.47) TRPA1MAPTCYP1A2CYP3A4CYP2D6
SCHEMBL28516934 0.79 TRPA1 (0.41) TRPA1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL17861316 0.79 CYP2A6 (0.53) TRPA1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL27978813 0.79 PLAU (0.51) MAPTCYP1A2CYP2C19CYP2A6MAP3K14
SCHEMBL26954239 0.79 CYP2A6 (0.44) MAPTCYP1A2CYP2A6TYMSTDP1
SCHEMBL30377849 0.75 CYP1A2 (0.52) CYP1A2CYP2A6TYMSCYP19A1CTDSP1
SCHEMBL8272301 0.75 TRPA1 (0.57) TRPA1MAPTCYP1A2CYP3A4CYP2D6
SCHEMBL28396185 0.75 TRPA1 (0.38) TRPA1CYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112358447-B Synthesis method of 7-fluoroisoquinoline-1-carboxylic acid 苏州康润医药有限公司 2022-04-12 CN disclosed
CN-112358447-A Synthesis method of 7-fluoroisoquinoline-1-carboxylic acid 苏州康润医药有限公司 2021-02-12 CN disclosed
CN-101228149-B Piperidinyl-substituted isoquinolinone derivatives as Rho-kinase inhibitors SANOFI AVENTIS 2013-01-02 CN disclosed