SCHEMBL28522683

SCHEMBL28522683

COc1ccc(NCC(=O)Oc2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.49
MAPT P10636 3/20 0.47
GAA P10253 2/20 0.47
CYP1A1 P04798 1/20 0.45
CYP1B1 Q16678 1/20 0.45
MAOB P27338 1/20 0.45
CTSL P07711 1/20 0.45
CTSS P25774 1/20 0.45
TP53 P04637 3/20 0.44
KMT2A Q03164 1/20 0.44
PTGDR2 Q9Y5Y4 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
KIF11 P52732 1/20 0.43
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43
ERBB2 P04626 1/20 0.43
PRKAB2 O43741 1/20 0.43
PRKAG1 P54619 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28523151 0.88 MAPT (0.55) POLBMAPTGAATP53KMT2A
SCHEMBL28531020 0.84 MAPT (0.51) POLBMAPTGAAMAOBKMT2A
SCHEMBL5112169 0.84 POLB (0.50) POLBKMT2AKIF11CA12CA1
SCHEMBL28516843 0.82 GAA (0.60) MAPTGAATP53KMT2ASMN1; SMN2
Hydrochloric Acid SCHEMBL5773679 0.82 POLB (0.49) POLBKMT2AKIF11CA12CA1
SCHEMBL28516840 0.81 MAPT (0.56) POLBMAPTGAAMAOBKMT2A
SCHEMBL28523007 0.81 KMT2A (0.59) MAPTGAATP53KMT2ASMN1; SMN2
SCHEMBL11665506 0.81 CYP1A1 (0.48) MAPTGAACYP1A1CYP1B1MAOB
SCHEMBL9779998 0.78 MAPT (0.59) POLBMAPTGAATP53KMT2A
SCHEMBL28528087 0.77 TP53 (0.52) MAPTGAATP53KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112279743-B Synthesis method of chiral alpha-amino acid ester derivative 中国科学院大连化学物理研究所 2022-10-18 CN disclosed
CN-112279743-A Synthesis method of chiral alpha-amino acid ester derivative 中国科学院大连化学物理研究所 2021-01-29 CN disclosed