SCHEMBL28523133

SCHEMBL28523133

Cc1ccc(N)cc1OCC(CC(=O)O)NC(=O)OC(C)(C)C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 7/20 0.50
ATM Q13315 1/20 0.38
SYK P43405 2/20 0.36
CTSS P25774 4/20 0.36
CTSK P43235 2/20 0.36
KLK5 Q9Y337 1/20 0.36
CYP2C9 P11712 1/20 0.36
HDAC3 O15379 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC10 Q969S8 1/20 0.35
HDAC11 Q96DB2 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
HDAC9 Q9UKV0 1/20 0.35
HDAC5 Q9UQL6 1/20 0.35
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18427975 1.00 AAK1 (0.50) AAK1ATMSYKCTSSCTSK
SCHEMBL28524725 0.91 AAK1 (0.58) AAK1ATMKLK5HDAC3HDAC4
SCHEMBL18428000 0.91 AAK1 (0.58) AAK1ATMKLK5HDAC3HDAC4
SCHEMBL18428059 0.83 AAK1 (0.47) AAK1
SCHEMBL18428103 0.82 ATM (0.42) AAK1ATMCTSSCTSKHDAC3
SCHEMBL28515403 0.82 ATM (0.42) AAK1ATMCTSSCTSKHDAC3
SCHEMBL23877853 0.82 ATM (0.42) AAK1ATMSYKCTSSCTSK
SCHEMBL16974957 0.82 ATM (0.42) AAK1ATMSYKCTSSCTSK
SCHEMBL16974958 0.82 ATM (0.42) AAK1ATMSYKCTSSCTSK
SCHEMBL18428084 0.81 F10 (0.49) AAK1ATMSYKKLK5HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108026026-B Beta-substituted beta-amino acids and analogs as chemotherapeutic agents and uses thereof 夸德里加生物科学公司 2021-02-09 CN disclosed