SCHEMBL28524725

SCHEMBL28524725

Cc1cc(N)ccc1OCC(CC(=O)O)NC(=O)OC(C)(C)C

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 12/20 0.58
ATM Q13315 1/20 0.38
ADRB2 P07550 1/20 0.36
ADRB1 P08588 1/20 0.36
ADRB3 P13945 1/20 0.36
HDAC3 O15379 2/20 0.36
HDAC4 P56524 2/20 0.36
HDAC1 Q13547 2/20 0.36
HDAC7 Q8WUI4 2/20 0.36
HDAC2 Q92769 2/20 0.36
HDAC10 Q969S8 2/20 0.36
HDAC11 Q96DB2 2/20 0.36
HDAC8 Q9BY41 2/20 0.36
HDAC6 Q9UBN7 2/20 0.36
HDAC9 Q9UKV0 2/20 0.36
HDAC5 Q9UQL6 2/20 0.36
KLK5 Q9Y337 1/20 0.36
PTGER1 P34995 1/20 0.36
TAS1R3 Q7RTX0 1/20 0.36
TAS1R1 Q7RTX1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18428000 1.00 AAK1 (0.58) AAK1ATMADRB2ADRB1ADRB3
SCHEMBL28523133 0.91 AAK1 (0.50) AAK1ATMHDAC3HDAC4HDAC1
SCHEMBL18427975 0.91 AAK1 (0.50) AAK1ATMHDAC3HDAC4HDAC1
SCHEMBL18428111 0.83 AAK1 (0.54) AAK1ADRB2ADRB1ADRB3
SCHEMBL28515403 0.82 ATM (0.42) AAK1ATMHDAC3HDAC4HDAC1
SCHEMBL18428103 0.82 ATM (0.42) AAK1ATMHDAC3HDAC4HDAC1
SCHEMBL28517888 0.81 F10 (0.49) AAK1ATMHDAC3HDAC4HDAC1
SCHEMBL18428084 0.81 F10 (0.49) AAK1ATMHDAC3HDAC4HDAC1
SCHEMBL18428005 0.81 AAK1 (0.52) AAK1ATMHDAC3HDAC4HDAC1
SCHEMBL16974966 0.81 ATM (0.46) AAK1ATMHDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108026026-B Beta-substituted beta-amino acids and analogs as chemotherapeutic agents and uses thereof 夸德里加生物科学公司 2021-02-09 CN disclosed