SCHEMBL28523368

SCHEMBL28523368

Cn1c(Cl)nc2[nH]ccc2c1=O

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.45
ADORA1 P30542 1/20 0.45
JAK2 O60674 2/20 0.41
JAK1 P23458 1/20 0.41
JAK3 P52333 1/20 0.41
DYRK1A Q13627 1/20 0.41
SIRT2 Q8IXJ6 1/20 0.40
RXFP1 Q9HBX9 1/20 0.38
PRKCI P41743 3/20 0.38
AXL P30530 2/20 0.38
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
TGFBR1 P36897 1/20 0.35
BRD4 O60885 1/20 0.35
TAF1 P21675 1/20 0.35
BRPF1 P55201 1/20 0.35
CREBBP Q92793 1/20 0.35
CECR2 Q9BXF3 1/20 0.35
BRD9 Q9H8M2 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12102100 0.81 ADORA2A (0.46) ADORA2AADORA1JAK2JAK1JAK3
SCHEMBL28510691 0.79 KDM4E (0.51) ADORA2AADORA1JAK2JAK1JAK3
SCHEMBL18321913 0.77 ADORA2A (0.42) ADORA2AADORA1JAK2JAK1JAK3
SCHEMBL28907542 0.73 JAK3 (0.43) ADORA2AADORA1JAK2JAK1JAK3
SCHEMBL29413023 0.72 KAT2B (0.49) BRD4TAF1BRPF1CREBBPCECR2
SCHEMBL28515190 0.72 ADORA2B (0.40) ADORA2AADORA1JAK2DYRK1ACYP1A2
SCHEMBL20894005 0.70 JAK2 (0.43) JAK2JAK1JAK3HRH4
SCHEMBL23505912 0.68 PRKCI (0.43) JAK2JAK1JAK3PRKCIAXL
SCHEMBL30879806 0.68 KDM4E (0.64) RXFP1SMN1; SMN2KDM4EALDH1A1MAPT
SCHEMBL2611507 0.68 KDM4E (0.64) RXFP1SMN1; SMN2KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107722013-B Deazapurine compounds, pharmaceutical compositions, preparation method and uses thereof 中国科学院上海药物研究所 2021-01-12 CN disclosed