SCHEMBL28524079

SCHEMBL28524079

O=C(O)Cc1cnc2ccc(Br)cc2n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.41
AURKB Q96GD4 2/20 0.41
KDR P35968 1/20 0.41
EGLN1 Q9GZT9 1/20 0.41
KDM4E B2RXH2 2/20 0.38
GLA P06280 1/20 0.38
MAPT P10636 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KMO O15229 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.37
ALDH1A1 P00352 3/20 0.37
GAA P10253 1/20 0.37
PDE10A Q9Y233 1/20 0.36
HDAC1 Q13547 2/20 0.36
HDAC2 Q92769 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
HTT P42858 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31193157 0.82 TSHR (0.43) KDM4EL3MBTL1ALDH1A1GAAHTT
SCHEMBL28500268 0.81 TLR9 (0.42) KDRKDM4EMAPTALDH1A1GAA
SCHEMBL30009200 0.79 BACE1 (0.46) AURKAAURKBKDREGLN1KDM4E
SCHEMBL25412037 0.78 PDE10A (0.60) KDM4EMAPTALDH1A1GAAPDE10A
SCHEMBL30134360 0.78 PDE10A (0.41) MAPTALDH1A1PDE10AMEN1KMT2A
SCHEMBL31043135 0.78 HTT (0.41) GLAPTGDR2ALDH1A1GAAHTT
SCHEMBL1641523 0.78 HDAC1 (0.52) AURKAAURKBKDREGLN1KDM4E
SCHEMBL17179171 0.77 HTT (0.41) MAPTALDH1A1PDE10AMEN1KMT2A
SCHEMBL23093834 0.77 PDE10A (0.40) MAPTALDH1A1PDE10AMEN1KMT2A
SCHEMBL30192121 0.77 PABPC1 (0.41) MAPTALDH1A1PDE10AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112125889-A Preparation method of 7-bromo-2- (1-methyl-1H-pyrazol-4-yl) quinoxaline 苏州明锐医药科技有限公司 2020-12-25 CN claimed