SCHEMBL28524718

SCHEMBL28524718

COc1ccc(N)c(OC(=O)CC(C)NC(=O)OC(C)(C)C)c1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 2/20 0.41
ABCB1 P08183 2/20 0.41
ALDH1A1 P00352 3/20 0.40
CYP3A4 P08684 1/20 0.40
CACNA1B Q00975 2/20 0.39
KDM4E B2RXH2 3/20 0.39
HPGD P15428 3/20 0.39
CYP2D6 P10635 1/20 0.39
PPARG P37231 1/20 0.39
PPARA Q07869 1/20 0.39
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
ACACB O00763 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28519457 0.91 AAK1 (0.41) AAK1ALDH1A1KDM4EHPGDCYP2D6
SCHEMBL28515407 0.89 AAK1 (0.39) AAK1ALDH1A1KDM4EHPGDCYP2D6
SCHEMBL28518871 0.85 AAK1 (0.41) AAK1ALDH1A1CYP2D6GAA
SCHEMBL28519453 0.85 AAK1 (0.41) AAK1ALDH1A1CACNA1BKDM4EHPGD
SCHEMBL28526489 0.84 AAK1 (0.41) AAK1CYP2D6PPARGPPARA
SCHEMBL28519422 0.82 CYP2D6 (0.43) AAK1CACNA1BCYP2D6PPARGPPARA
SCHEMBL28521318 0.81 KDM4E (0.40) AAK1ALDH1A1CACNA1BKDM4ECYP2D6
SCHEMBL28520580 0.77 CYP2D6 (0.40) AAK1ALDH1A1KDM4EHPGDCYP2D6
SCHEMBL28515363 0.77 CYP2D6 (0.40) AAK1ALDH1A1CACNA1BKDM4EHPGD
SCHEMBL15964931 0.76 PPARA (0.49) AAK1ALDH1A1CYP3A4CACNA1BPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108026026-B Beta-substituted beta-amino acids and analogs as chemotherapeutic agents and uses thereof 夸德里加生物科学公司 2021-02-09 CN disclosed