SCHEMBL28520580

SCHEMBL28520580

Cc1ccc(N)cc1OC(=O)CC(C)NC(=O)OC(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.40
AAK1 Q2M2I8 6/20 0.40
MAPT P10636 4/20 0.38
HPGD P15428 4/20 0.38
ALDH1A1 P00352 3/20 0.38
TSHR P16473 2/20 0.38
CA2 P00918 3/20 0.38
CA1 P00915 2/20 0.38
CA7 P43166 2/20 0.38
CA4 P22748 1/20 0.38
CA9 Q16790 1/20 0.38
LMNA P02545 2/20 0.37
HSD17B10 Q99714 2/20 0.37
KDM4E B2RXH2 2/20 0.37
GAA P10253 2/20 0.37
GLA P06280 1/20 0.37
CASP1 P29466 1/20 0.37
RAB9A P51151 1/20 0.37
CASP7 P55210 1/20 0.37
ALOX5 P09917 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28521318 0.87 KDM4E (0.40) CYP2D6AAK1ALDH1A1CA2CA1
SCHEMBL28448730 0.85 AAK1 (0.41) CYP2D6AAK1MAPTHPGDALDH1A1
SCHEMBL61961 0.84 ALDH1A1 (0.52) CYP2D6AAK1MAPTHPGDALDH1A1
SCHEMBL28515363 0.81 CYP2D6 (0.40) CYP2D6AAK1MAPTHPGDALDH1A1
SCHEMBL28519422 0.79 CYP2D6 (0.43) CYP2D6AAK1CA2CA1CA7
SCHEMBL28519453 0.78 AAK1 (0.41) CYP2D6AAK1MAPTHPGDALDH1A1
SCHEMBL28518871 0.78 AAK1 (0.41) CYP2D6AAK1ALDH1A1CA2CA1
SCHEMBL28519457 0.77 AAK1 (0.41) CYP2D6AAK1MAPTHPGDALDH1A1
SCHEMBL28524718 0.77 AAK1 (0.41) CYP2D6AAK1MAPTHPGDALDH1A1
SCHEMBL28526489 0.77 AAK1 (0.41) CYP2D6AAK1CA2CA1CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108026026-B Beta-substituted beta-amino acids and analogs as chemotherapeutic agents and uses thereof 夸德里加生物科学公司 2021-02-09 CN disclosed