SCHEMBL28524858

SCHEMBL28524858

NC(=O)O[C@H]1C[C@@H](Nc2cnc(C(F)(F)F)cn2)C1

nearest known ligand 0.43

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 18/20 0.43
CCNK O75909 1/20 0.42
CDK12 Q9NYV4 1/20 0.42
HCRTR2 O43614 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21491972 0.78 HCRTR1 (0.44) HCRTR1CCNKCDK12
SCHEMBL30744401 0.78 HCRTR1 (0.44) HCRTR1CCNKCDK12
SCHEMBL21491975 0.78 HCRTR1 (0.44) HCRTR1CCNKCDK12
SCHEMBL21492759 0.77 HCRTR1 (0.48) HCRTR1CCNKCDK12HCRTR2
Hydrochloric Acid SCHEMBL21491930 0.76 HCRTR1 (0.43) HCRTR1CCNKCDK12
Hydrochloric Acid SCHEMBL30744328 0.76 HCRTR1 (0.43) HCRTR1CCNKCDK12
Hydrochloric Acid SCHEMBL21491928 0.76 HCRTR1 (0.43) HCRTR1CCNKCDK12
SCHEMBL30744422 0.74 HCRTR1 (0.45) HCRTR1CCNKCDK12
SCHEMBL21503414 0.74 HCRTR1 (0.45) HCRTR1CCNKCDK12
SCHEMBL26693505 0.74 HCRTR1 (0.45) HCRTR1CCNKCDK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112218865-B Pteridinone compounds and uses thereof 沃泰克斯药物股份有限公司 2024-03-12 CN disclosed
CN-112218865-A Pteridinone compounds and uses thereof 沃泰克斯药物股份有限公司 2021-01-12 CN disclosed