SCHEMBL28525698

SCHEMBL28525698

COC(=O)c1cc(F)ncc1C.Cc1cnc(F)cc1I

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 1/20 0.38
SOS1 Q07889 1/20 0.36
ATM Q13315 1/20 0.34
NPC1 O15118 1/20 0.34
CASP3 P42574 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
SENP8 Q96LD8 1/20 0.34
SENP7 Q9BQF6 1/20 0.34
SENP6 Q9GZR1 1/20 0.34
TSHR P16473 2/20 0.33
NQO2 P16083 1/20 0.33
KMT2A Q03164 1/20 0.33
NR4A2 P43354 1/20 0.33
KDM4E B2RXH2 3/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
MAPT P10636 2/20 0.33
MAPK1 P28482 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GLA P06280 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19641106 0.91 ATM (0.40) ATMNPC1CASP3RAB9ASMN1; SMN2
SCHEMBL363228 0.79
SCHEMBL29823074 0.79
SCHEMBL20951861 0.78 NNMT (0.44) ATMNPC1CASP3RAB9ASMN1; SMN2
SCHEMBL29878684 0.74 MAPK1 (0.47) ATMKDM4EL3MBTL1MAPTMAPK1
SCHEMBL9641326 0.74 ATM (0.42) ATMTSHRKMT2ANR4A2KDM4E
SCHEMBL17490653 0.74 KDM4E (0.44) ATMTSHRKMT2ANR4A2KDM4E
SCHEMBL21232045 0.73 KDM4E (0.51) CFTRATMTSHRNQO2KDM4E
SCHEMBL29574200 0.73 SOS1 (0.43) SOS1TSHRKMT2ANR4A2KDM4E
SCHEMBL17558778 0.73 SOS1 (0.43) SOS1TSHRKMT2ANR4A2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112351780-B Substituted heterocyclic inhibitors of PTPN11 纳维尔制药有限公司 2023-12-01 CN disclosed
CN-112351780-A Substituted heterocyclic inhibitors of PTPN11 纳维尔制药有限公司 2021-02-09 CN disclosed