SCHEMBL28525810

SCHEMBL28525810

O=C1NC2(CCCCC2)Oc2ccc([N+](=O)[O-])cc21

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.58
CNR2 P34972 1/20 0.49
CYP3A4 P08684 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
CAPN9 O14815 1/20 0.43
CASP3 P42574 1/20 0.43
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
TDP2 O95551 1/20 0.41
HDAC3 O15379 2/20 0.41
HDAC4 P56524 2/20 0.41
HDAC1 Q13547 2/20 0.41
HDAC7 Q8WUI4 2/20 0.41
HDAC2 Q92769 2/20 0.41
HDAC10 Q969S8 2/20 0.41
HDAC11 Q96DB2 2/20 0.41
HDAC8 Q9BY41 2/20 0.41
HDAC6 Q9UBN7 2/20 0.41
HDAC9 Q9UKV0 2/20 0.41
HDAC5 Q9UQL6 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28525814 0.99 ALDH1A1 (0.56) ALDH1A1CNR2CYP3A4TDP1CAPN9
SCHEMBL28524830 0.79 CYP3A4 (0.53) ALDH1A1CYP3A4TDP1CAPN9CASP3
SCHEMBL29634212 0.79 CYP3A4 (0.53) ALDH1A1CYP3A4TDP1CAPN9CASP3
SCHEMBL28523381 0.78 ALDH1A1 (0.64) ALDH1A1CNR2TDP1MEN1KMT2A
SCHEMBL29770999 0.76 ALDH1A1 (0.61) ALDH1A1CNR2TDP1MEN1KMT2A
SCHEMBL8130642 0.75 CYP3A4 (0.48) ALDH1A1CYP3A4TDP1CAPN9CASP3
SCHEMBL28520051 0.75 CYP3A4 (0.48) ALDH1A1CYP3A4TDP1CAPN9CASP3
SCHEMBL29634204 0.75 CYP3A4 (0.48) ALDH1A1CYP3A4TDP1CAPN9CASP3
SCHEMBL11103515 0.75 KDM4E (0.63) ALDH1A1CYP3A4TDP1MEN1KMT2A
SCHEMBL7508014 0.74 ALDH1A1 (1.00) ALDH1A1CNR2TDP1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022160138-A1 BENZOXAZINE-4-ONE COMPOUND, PREPARATION METHOD THEREFOR, AND MEDICAL USE THEREOF 承德医学院 2022-08-04 WO disclosed
CN-112442022-B Benzoxazine-4-ketone compound, preparation method and medical application thereof 承德医学院 2022-05-20 CN disclosed
CN-112442022-A Benzoxazine-4-ketone compound, preparation method and medical application thereof 承德医学院 2021-03-05 CN disclosed