SCHEMBL28525906

SCHEMBL28525906

CC(Nc1ncc2ccc(=O)n(C)c2n1)c1ccc(C(=O)O)cc1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 6/20 0.52
CCND1 P24385 6/20 0.52
CCND2 P30279 6/20 0.52
CCND3 P30281 6/20 0.52
MAPK8 P45983 2/20 0.48
MAPK9 P45984 1/20 0.48
MAPK10 P53779 1/20 0.48
HDAC3 O15379 4/20 0.42
HDAC1 Q13547 4/20 0.42
HDAC2 Q92769 4/20 0.42
HDAC6 Q9UBN7 4/20 0.42
LDHA P00338 1/20 0.41
LDHB P07195 1/20 0.41
PTK2 Q05397 1/20 0.40
FGFR1 P11362 1/20 0.40
PHGDH O43175 3/20 0.39
VNN1 O95497 1/20 0.39
GSK3A P49840 1/20 0.39
GSK3B P49841 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28525903 1.00 CDK4 (0.52) CDK4CCND1CCND2CCND3MAPK8
SCHEMBL23141677 0.89 CDK4 (0.47) CDK4CCND1CCND2CCND3MAPK8
SCHEMBL23141676 0.89 CDK4 (0.47) CDK4CCND1CCND2CCND3MAPK8
SCHEMBL28537531 0.86 CDK4 (0.69) CDK4CCND1CCND2CCND3MAPK8
SCHEMBL28537530 0.86 CDK4 (0.69) CDK4CCND1CCND2CCND3MAPK8
SCHEMBL28909366 0.82 CDK4 (0.58) CDK4CCND1CCND2CCND3MAPK8
SCHEMBL28909368 0.82 CDK4 (0.58) CDK4CCND1CCND2CCND3MAPK8
SCHEMBL5265689 0.81 CDK4 (0.68) CDK4CCND1CCND2CCND3MAPK8
SCHEMBL23141494 0.79 CDK4 (0.49) CDK4CCND1CCND2CCND3MAPK8
SCHEMBL23141496 0.79 CDK4 (0.49) CDK4CCND1CCND2CCND3MAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112469719-A Heterocondensed pyridone compounds and their use as IDH inhibitors 内尔维亚诺医疗科学公司 2021-03-09 CN claimed
CN-112469719-A Heterocondensed pyridone compounds and their use as IDH inhibitors 内尔维亚诺医疗科学公司 2021-03-09 CN disclosed