SCHEMBL28526280

SCHEMBL28526280

CN1CCCC(c2ccccc2C2CCCN2)C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.43
KCNH2 Q12809 2/20 0.43
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
DRD3 P35462 2/20 0.43
KDM4E B2RXH2 1/20 0.42
ATM Q13315 1/20 0.42
TAAR1 Q96RJ0 1/20 0.41
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
CYP2D6 P10635 1/20 0.40
TSHR P16473 1/20 0.40
CHRM2 P08172 1/20 0.40
HTR1A P08908 1/20 0.40
ADRA2A P08913 1/20 0.40
CHRM1 P11229 1/20 0.40
DRD1 P21728 1/20 0.40
TBXA2R P21731 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23487422 0.93 KDM4E (0.49) KDM4EATMTAAR1CHRM2CHRM1
SCHEMBL28527428 0.84 TAAR1 (0.43) HTR2AKDM4EATMTAAR1CHRM2
SCHEMBL28527431 0.84 TAAR1 (0.43) HTR2AKDM4EATMTAAR1CHRM2
SCHEMBL28537464 0.84 TAAR1 (0.43) HTR2AKDM4EATMTAAR1CHRM2
SCHEMBL28526313 0.80 CHRM5 (0.44) HTR2CTAAR1CYP2D6CHRM2CHRM1
SCHEMBL24737035 0.80 CHRM5 (0.44) HTR2CTAAR1CYP2D6CHRM2CHRM1
SCHEMBL28527595 0.78 CHRM5 (0.43) HTR2CTAAR1CYP2D6CHRM2CHRM1
SCHEMBL23323069 0.78 CHRM5 (0.46) HTR2CTAAR1CYP2D6CHRM2CHRM1
SCHEMBL22165432 0.78 CHRM5 (0.46) HTR2CTAAR1CYP2D6CHRM2CHRM1
SCHEMBL22165430 0.78 CHRM5 (0.46) HTR2CTAAR1CYP2D6CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117683029-A Bcl-2 inhibitors 百济神州有限公司 2024-03-12 CN disclosed
CN-112437772-B Bcl-2 inhibitors 百济神州有限公司 2023-11-21 CN disclosed
CN-112437772-A Bcl-2 inhibitors 百济神州有限公司 2021-03-02 CN disclosed