SCHEMBL28526304

SCHEMBL28526304

CN(C)C1C[C@H](c2ccccc2C2CCCN2c2ccc(Br)cc2)CCN1

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.32
HTR2A P28223 2/20 0.32
HTR2C P28335 2/20 0.32
HTR2B P41595 2/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
MAPK1 P28482 1/20 0.32
CYP2C19 P33261 1/20 0.32
PIK3CB P42338 1/20 0.31
NOS1 P29475 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28534516 0.83 PIK3CB (0.35) CYP2D6CYP2C9MAPK1CYP2C19PIK3CB
SCHEMBL31525091 0.81 HTR2C (0.41) HTR2CHTR2BCYP2D6CYP2C9MAPK1
SCHEMBL28529794 0.81 HTR2C (0.41) HTR2CHTR2BCYP2D6CYP2C9MAPK1
SCHEMBL28529792 0.81 HTR2C (0.41) HTR2CHTR2BCYP2D6CYP2C9MAPK1
SCHEMBL28528284 0.79 CYP2D6 (0.38) HRH3CYP2D6CYP2C9MAPK1CYP2C19
SCHEMBL28528279 0.79 CYP2D6 (0.38) HRH3CYP2D6CYP2C9MAPK1CYP2C19
SCHEMBL28909552 0.76 HRH3 (0.41) HRH3HTR2BCYP2D6CYP2C9MAPK1
SCHEMBL28909558 0.76 HRH3 (0.41) HRH3HTR2BCYP2D6CYP2C9MAPK1
SCHEMBL24775580 0.75 HRH3 (0.38) HRH3CYP2D6CYP2C9MAPK1CYP2C19
SCHEMBL28532862 0.70 MAPT (0.41) CYP2D6CYP2C9MAPK1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117683029-A Bcl-2 inhibitors 百济神州有限公司 2024-03-12 CN disclosed
CN-117430601-A Bcl-2 inhibitors 百济神州有限公司 2024-01-23 CN disclosed
CN-112437772-B Bcl-2 inhibitors 百济神州有限公司 2023-11-21 CN disclosed
CN-112437772-A Bcl-2 inhibitors 百济神州有限公司 2021-03-02 CN disclosed