SCHEMBL28526454

SCHEMBL28526454

Cc1ccc(N)cc1C(=O)C[C@@H](CC(=O)OC(C)(C)C)NC(=O)OC(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.41
AAK1 Q2M2I8 4/20 0.39
ATM Q13315 1/20 0.37
ALDH1A1 P00352 4/20 0.36
MAPT P10636 4/20 0.36
HPGD P15428 2/20 0.36
KDM4E B2RXH2 1/20 0.36
GAA P10253 1/20 0.36
PKM P14618 1/20 0.36
ALOX12 P18054 1/20 0.36
ALOX5 P09917 1/20 0.35
SYK P43405 1/20 0.35
ADRB2 P07550 1/20 0.35
ADRB1 P08588 1/20 0.35
ADRB3 P13945 1/20 0.35
TSHR P16473 1/20 0.35
KLK5 Q9Y337 1/20 0.34
BRD4 O60885 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28526456 1.00 CYP2D6 (0.41) CYP2D6AAK1ATMALDH1A1MAPT
SCHEMBL28859563 0.91 AAK1 (0.39) AAK1ATMALDH1A1MAPTHPGD
SCHEMBL18428123 0.91 AAK1 (0.39) AAK1ATMALDH1A1MAPTHPGD
SCHEMBL18472360 0.84 ADRB2 (0.36) CYP2D6AAK1ALDH1A1MAPTHPGD
SCHEMBL28520956 0.83 CYP2D6 (0.42) CYP2D6AAK1ATMALDH1A1MAPT
SCHEMBL16970672 0.83 CYP2D6 (0.42) CYP2D6AAK1ATMALDH1A1MAPT
SCHEMBL28520959 0.83 CYP2D6 (0.42) CYP2D6AAK1ATMALDH1A1MAPT
SCHEMBL28526994 0.83 KMT2A (0.42) CYP2D6ALDH1A1MAPTHPGDGAA
SCHEMBL28526991 0.83 KMT2A (0.42) CYP2D6ALDH1A1MAPTHPGDGAA
SCHEMBL28907010 0.81 CYP2D6 (0.41) CYP2D6AAK1ATMALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108026026-B Beta-substituted beta-amino acids and analogs as chemotherapeutic agents and uses thereof 夸德里加生物科学公司 2021-02-09 CN disclosed