SCHEMBL28527342

SCHEMBL28527342

Cc1c(O)ccc2c1cc1n2CCC1CC(=O)O

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 17/20 0.42
S1PR5 Q9H228 3/20 0.40
S1PR4 O95977 1/20 0.39
TBXA2R P21731 2/20 0.37
PTGDR Q13258 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2018070 0.86 GAA (0.37) S1PR1
SCHEMBL28537384 0.85 S1PR1 (0.52) S1PR1S1PR5S1PR4
SCHEMBL12320295 0.75 S1PR1 (0.54) S1PR1S1PR5S1PR4
SCHEMBL2016037 0.75 S1PR1 (0.54) S1PR1S1PR5S1PR4
SCHEMBL2923853 0.74 PTGDR (0.53) S1PR1S1PR5TBXA2RPTGDRPTGDR2
SCHEMBL2922357 0.74 PTGDR (0.44) S1PR1TBXA2RPTGDRPTGDR2
SCHEMBL5775673 0.73 S1PR1 (0.42) S1PR1S1PR5S1PR4TBXA2RPTGDR
SCHEMBL2016666 0.73 S1PR1 (0.41) S1PR1S1PR5
SCHEMBL2926749 0.73 TBXA2R (0.54) S1PR1TBXA2RPTGDRPTGDR2
SCHEMBL5778068 0.72 TBXA2R (0.44) S1PR1S1PR5TBXA2RPTGDRPTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105816453-B Substituted tricyclic acid derivatives as S1P1 receptor agonists for the treatment of autoimmune and inflammatory disorders 艾尼纳制药公司 2021-03-05 CN disclosed