SCHEMBL28537384

SCHEMBL28537384

COc1ccc2c(cc3n2CCC3CC(=O)O)c1C

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 19/20 0.52
S1PR5 Q9H228 4/20 0.44
S1PR4 O95977 3/20 0.40
CYP2C9 P11712 1/20 0.39
FFAR4 Q5NUL3 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2016666 0.87 S1PR1 (0.41) S1PR1S1PR5
SCHEMBL28527342 0.85 S1PR1 (0.42) S1PR1S1PR5S1PR4
SCHEMBL2021001 0.76 S1PR1 (0.75) S1PR1S1PR5S1PR4CYP2C9
SCHEMBL2016746 0.76 S1PR1 (0.75) S1PR1S1PR5S1PR4CYP2C9
SCHEMBL2016745 0.76 S1PR1 (0.75) S1PR1S1PR5S1PR4CYP2C9
SCHEMBL17690538 0.76 S1PR1 (0.62) S1PR1S1PR5S1PR4CYP2C9
SCHEMBL5775625 0.75 S1PR1 (0.47) S1PR1S1PR5S1PR4FFAR4
SCHEMBL2018070 0.74 GAA (0.37) S1PR1
SCHEMBL2923853 0.72 PTGDR (0.53) S1PR1S1PR5
SCHEMBL2922357 0.72 PTGDR (0.44) S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105816453-B Substituted tricyclic acid derivatives as S1P1 receptor agonists for the treatment of autoimmune and inflammatory disorders 艾尼纳制药公司 2021-03-05 CN disclosed