SCHEMBL28529048

SCHEMBL28529048

NC(=O)c1ccc2ccnccc1-2

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHUK O15111 4/20 0.56
IKBKB O14920 4/20 0.53
BCAT2 O15382 1/20 0.52
CASP1 P29466 1/20 0.51
IKBKE Q14164 2/20 0.51
PKMYT1 Q99640 1/20 0.51
CDC7 O00311 5/20 0.50
CDK9 P50750 1/20 0.50
BTK Q06187 2/20 0.49
CCNC P24863 4/20 0.49
CDK8 P49336 4/20 0.49
SIRT3 Q9NTG7 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
ROCK2 O75116 1/20 0.47
MAP4K4 O95819 1/20 0.47
GSK3B P49841 1/20 0.47
CLK4 Q9HAZ1 1/20 0.47
MKNK2 Q9HBH9 1/20 0.47
CHEK2 O96017 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6448102 0.87 BCAT2 (0.67) CHUKIKBKBBCAT2CASP1IKBKE
SCHEMBL25306948 0.86 SIRT3 (0.61) CHUKIKBKBBCAT2CASP1IKBKE
SCHEMBL164881 0.86 BCAT2 (0.71) CHUKIKBKBBCAT2CASP1IKBKE
Hydrochloric Acid SCHEMBL4597839 0.85 BCAT2 (0.69) CHUKIKBKBBCAT2CASP1IKBKE
Hydrochloric Acid SCHEMBL29710331 0.85 BCAT2 (0.69) CHUKIKBKBBCAT2CASP1IKBKE
Hydrochloric Acid SCHEMBL9027847 0.85 BCAT2 (0.69) CHUKIKBKBBCAT2CASP1IKBKE
SCHEMBL28829405 0.82 CHEK2 (0.52) CHUKIKBKBCASP1IKBKEPKMYT1
SCHEMBL27193217 0.80 CHUK (0.61) CHUKIKBKBCASP1IKBKEPKMYT1
SCHEMBL27193240 0.79 CHUK (0.55) CHUKIKBKBCASP1IKBKEPKMYT1
SCHEMBL27996934 0.78 CCNC (0.55) CHUKIKBKBCASP1IKBKEPKMYT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117729916-A Benzodioxane modulators of leukotriene A4 hydrolase (LTA 4H) for the prevention and treatment of aging-related diseases 万能溶剂有限公司 2024-03-19 CN claimed
CN-112469439-A With leukotriene A4Hydrolase modulators for the treatment of aging-related diseases 万能溶剂有限公司 2021-03-09 CN disclosed