SCHEMBL28529940

SCHEMBL28529940

Cc1ccc2nc(-c3ccccc3)c(C)cc2c1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.73
KDM4E B2RXH2 4/20 0.68
ALDH1A1 P00352 2/20 0.68
L3MBTL1 Q9Y468 1/20 0.68
PSMB5 P28074 2/20 0.62
TDP1 Q9NUW8 1/20 0.56
MAPT P10636 3/20 0.54
LMNA P02545 2/20 0.54
DHODH Q02127 1/20 0.50
NPC1 O15118 1/20 0.47
POLB P06746 1/20 0.47
HPGD P15428 1/20 0.47
CASP3 P42574 1/20 0.47
RAB9A P51151 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
SENP8 Q96LD8 1/20 0.47
SENP7 Q9BQF6 1/20 0.47
SENP6 Q9GZR1 1/20 0.47
NQO2 P16083 1/20 0.47
KLK7 P49862 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4143806 0.89 PDE10A (0.56) PDE10AKDM4EALDH1A1L3MBTL1PSMB5
SCHEMBL28528610 0.87 PDE10A (0.71) PDE10AKDM4EALDH1A1L3MBTL1PSMB5
SCHEMBL3842193 0.87 PDE10A (0.56) PDE10AKDM4EALDH1A1L3MBTL1PSMB5
SCHEMBL28893755 0.86 KDM4E (0.64) PDE10AKDM4EALDH1A1L3MBTL1PSMB5
SCHEMBL2125225 0.85 PDE10A (1.00) PDE10AKDM4EALDH1A1L3MBTL1PSMB5
SCHEMBL17942681 0.84 KDM4E (0.62) PDE10AKDM4EALDH1A1L3MBTL1PSMB5
SCHEMBL6858227 0.83 PDE10A (0.96) PDE10AKDM4EALDH1A1L3MBTL1PSMB5
SCHEMBL27610987 0.83 PDE10A (0.96) PDE10AKDM4EALDH1A1L3MBTL1PSMB5
SCHEMBL30999690 0.83 PDE10A (0.96) PDE10AKDM4EALDH1A1L3MBTL1PSMB5
SCHEMBL4097200 0.83 PDE10A (0.50) PDE10AKDM4EALDH1A1L3MBTL1PSMB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112521333-A Synthesis method of chiral 2, 3-disubstituted tetrahydroquinoline derivative 中国科学院大连化学物理研究所 2021-03-19 CN disclosed