SCHEMBL28530232

SCHEMBL28530232

CC12CC3CC(C1)CC(C)(C3)C2.O=C(Nc1nc2ccc(OC(F)(F)F)cc2s1)C12CC3CC(CC(C3)C1)C2

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.59
RAB9A P51151 3/20 0.59
DYRK1A Q13627 2/20 0.58
CNR1 P21554 1/20 0.54
CSNK1D P48730 4/20 0.49
CLK1 P49759 1/20 0.49
KCNQ3 O43525 1/20 0.49
KCNQ2 O43526 1/20 0.49
HDAC3 O15379 1/20 0.49
HDAC4 P56524 1/20 0.49
HDAC1 Q13547 1/20 0.49
HDAC7 Q8WUI4 1/20 0.49
HDAC2 Q92769 1/20 0.49
HDAC10 Q969S8 1/20 0.49
HDAC11 Q96DB2 1/20 0.49
HDAC8 Q9BY41 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
HDAC9 Q9UKV0 1/20 0.49
HDAC5 Q9UQL6 1/20 0.49
ACP1 P24666 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30944320 0.93 DYRK1A (0.64) NPC1RAB9ADYRK1ACNR1CSNK1D
SCHEMBL31236386 0.91 DYRK1A (0.60) NPC1RAB9ADYRK1ACNR1CSNK1D
SCHEMBL28518076 0.91 DYRK1A (0.60) NPC1RAB9ADYRK1ACNR1CSNK1D
SCHEMBL28520293 0.85 DYRK1A (0.62) NPC1RAB9ADYRK1ACNR1CSNK1D
SCHEMBL30944290 0.85 DYRK1A (0.62) NPC1RAB9ADYRK1ACNR1CSNK1D
SCHEMBL30444394 0.82 DYRK1A (0.61) NPC1RAB9ADYRK1ACNR1CSNK1D
SCHEMBL30944323 0.82 CNR1 (0.64) NPC1RAB9ADYRK1ACNR1CSNK1D
SCHEMBL28527319 0.82 CNR1 (0.64) NPC1RAB9ADYRK1ACNR1CSNK1D
SCHEMBL4920969 0.82 NPC1 (0.75) NPC1RAB9ADYRK1ACNR1CSNK1D
SCHEMBL30944325 0.81 DYRK1A (0.65) NPC1RAB9ADYRK1ACSNK1DHDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112423746-A Novel anti-mycobacterial heterocyclic amides 克莱斯通公司 2021-02-26 CN claimed