SCHEMBL28530643

SCHEMBL28530643

Cc1ccnc(C(C)C)c1Nc1cc(Cl)nc(Cl)c1C(N)=O

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.38
MAPT P10636 1/20 0.35
ALDH1A1 P00352 3/20 0.34
HPGD P15428 2/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
GAA P10253 1/20 0.34
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
SYK P43405 3/20 0.33
KCNH2 Q12809 1/20 0.33
HTT P42858 1/20 0.33
TDO2 P48775 1/20 0.32
TAAR1 Q96RJ0 1/20 0.32
KRAS P01116 1/20 0.32
TP53 P04637 1/20 0.32
BLM P54132 1/20 0.32
CISD2 Q8N5K1 1/20 0.32
CLCN2 P51788 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30544155 1.00 POLB (0.38) POLBMAPTALDH1A1HPGDRAB9A
SCHEMBL28661419 0.83 MAPT (0.42) POLBMAPTALDH1A1HPGDRAB9A
SCHEMBL29427867 0.83 MAPT (0.42) POLBMAPTALDH1A1HPGDRAB9A
SCHEMBL29427882 0.80 KRAS (0.33) MAPTALDH1A1HPGDRAB9ASMN1; SMN2
SCHEMBL22623071 0.80 KRAS (0.33) MAPTALDH1A1HPGDRAB9ASMN1; SMN2
SCHEMBL24069476 0.75 CLCN2 (0.37) MAPTALDH1A1RAB9ASMN1; SMN2GAA
SCHEMBL30106566 0.75 CLCN2 (0.37) MAPTALDH1A1RAB9ASMN1; SMN2GAA
SCHEMBL29427879 0.75 CLCN2 (0.51) CLCN2
SCHEMBL28783719 0.74 POLB (0.35) POLBKRAS
SCHEMBL31361068 0.74 ALDH1A1 (0.44) POLBMAPTALDH1A1HPGDRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112390818-B Substituted heteroaromatic dihydro pyrimidinone derivatives, their preparation and pharmaceutical use 劲方医药科技(上海)有限公司 2023-08-22 CN disclosed
CN-112390818-A Substituted heteroaromatic dihydro pyrimidone derivatives, preparation method and medical application thereof 劲方医药科技(上海)有限公司 2021-02-23 CN disclosed