SCHEMBL28533456

SCHEMBL28533456

O=C1NCCc2cc(C3=CCNCC3)c(-n3cnc(C4CC4)c3)cc21

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 7/20 0.36
KDM4E B2RXH2 1/20 0.32
GSK3B P49841 1/20 0.31
GRM5 P41594 2/20 0.31
GRM1 Q13255 1/20 0.31
MAPK1 P28482 1/20 0.31
PARP10 Q53GL7 6/20 0.30
PARP1 P09874 4/20 0.30
PARP11 Q9NR21 2/20 0.30
F7 P08709 1/20 0.30
F3 P13726 1/20 0.30
HTR6 P50406 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28539135 0.83 MAP3K5 (0.38) MAP3K5GSK3BGRM5GRM1PARP10
SCHEMBL28541383 0.81 MAP3K5 (0.35) MAP3K5GSK3BGRM5GRM1
SCHEMBL28607413 0.81 MAP3K5 (0.38) MAP3K5KDM4EGSK3BGRM5GRM1
SCHEMBL22473965 0.81 PARP10 (0.41) MAP3K5KDM4EGSK3BGRM5GRM1
SCHEMBL28941273 0.80 PARP10 (0.40) MAP3K5KDM4EGRM5GRM1PARP10
SCHEMBL28887761 0.80 PARP10 (0.40) MAP3K5KDM4EGSK3BGRM5GRM1
SCHEMBL20489212 0.80 MAP3K5 (0.49) MAP3K5KDM4EPARP10PARP1PARP11
SCHEMBL29978642 0.80 MAP3K5 (0.49) MAP3K5KDM4EPARP10PARP1PARP11
SCHEMBL30362996 0.80 PARP10 (0.40) MAP3K5KDM4EGRM5GRM1PARP10
SCHEMBL28910942 0.76 MAP3K5 (0.39) MAP3K5KDM4EGSK3BGRM5GRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109071498-B Kinase inhibitor and preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2021-03-30 CN disclosed