SCHEMBL28534402

SCHEMBL28534402

COS(=O)(=O)CC1(c2ccc(Cl)cc2Cl)CC1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 5/20 0.47
SLC6A4 P31645 4/20 0.47
CYP3A4 P08684 1/20 0.34
MAPT P10636 2/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
POLB P06746 1/20 0.34
HPGD P15428 1/20 0.34
RAB9A P51151 1/20 0.34
KMT2A Q03164 1/20 0.34
SLC6A2 P23975 1/20 0.34
GRM5 P41594 1/20 0.34
TRPV4 Q9HBA0 1/20 0.33
RORC P51449 1/20 0.33
PTGS2 P35354 1/20 0.33
HSD11B1 P28845 1/20 0.32
HSD11B2 P80365 1/20 0.32
DPP4 P27487 1/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28534405 0.72 SLC6A3 (0.41) SLC6A3SLC6A4CYP3A4MAPTKMT2A
SCHEMBL9481114 0.71 SLC6A3 (0.55) SLC6A3SLC6A4CYP3A4ALDH1A1SLC6A2
SCHEMBL21723004 0.71 SLC6A4 (0.57) SLC6A3SLC6A4SLC6A2GRM5HSD11B1
SCHEMBL17761221 0.68 SLC6A3 (0.54) SLC6A3SLC6A4CYP3A4MAPTKDM4E
SCHEMBL27355315 0.65 POLB (0.40) SLC6A4KDM4EALDH1A1POLBHPGD
SCHEMBL9481251 0.65 SLC6A4 (0.68) SLC6A3SLC6A4SLC6A2
SCHEMBL20978149 0.65 SLC6A4 (0.50) SLC6A3SLC6A4SLC6A2
SCHEMBL9921757 0.64 SLC6A3 (0.49) SLC6A3SLC6A4CYP3A4MAPTSLC6A2
SCHEMBL3517321 0.64 SLC6A3 (1.00) SLC6A3SLC6A4SLC6A2DPP4
SCHEMBL3520534 0.64 SLC6A4 (1.00) SLC6A3SLC6A4SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112867720-A Novel heterocyclic compounds as monoacylglycerol lipase inhibitors 豪夫迈·罗氏有限公司 2021-05-28 CN disclosed
CN-112469724-A Novel heterocyclic compounds as monoacylglycerol lipase inhibitors 豪夫迈·罗氏有限公司 2021-03-09 CN disclosed