SCHEMBL28535010

SCHEMBL28535010

O=C(Cl)c1c(F)cc(-c2ccccc2)cc1F.O=C(O)c1c(F)cc(-c2ccccc2)cc1F

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C2 P52895 3/20 0.53
AKR1C1 Q04828 3/20 0.53
DHODH Q02127 6/20 0.42
ALDH1A1 P00352 1/20 0.41
ALOX15 P16050 1/20 0.41
RHEB Q15382 1/20 0.40
EGFR P00533 1/20 0.40
KMO O15229 1/20 0.39
PTPN1 P18031 1/20 0.39
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
HSD17B10 Q99714 1/20 0.39
AKR1C4 P17516 1/20 0.38
AKR1C3 P42330 1/20 0.38
ACLY P53396 1/20 0.37
ERN1 O75460 1/20 0.37
DHFR P00374 1/20 0.37
HNF4A P41235 1/20 0.37
MCL1 Q07820 1/20 0.37
ACMSD Q8TDX5 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17848889 0.94 AKR1C2 (0.53) AKR1C2AKR1C1DHODHALDH1A1ALOX15
SCHEMBL505832 0.91 AKR1C2 (0.61) AKR1C2AKR1C1DHODHALDH1A1EGFR
Biphenyl SCHEMBL2838517 0.81 AKR1C2 (0.50) AKR1C2AKR1C1DHODHALDH1A1KMO
SCHEMBL28888036 0.80 AKR1C2 (0.45) AKR1C2AKR1C1ALDH1A1KMOKDM4E
SCHEMBL10029672 0.79 AKR1C2 (0.56) AKR1C2AKR1C1DHODHALDH1A1EGFR
SCHEMBL28138125 0.79 CES2 (0.54) ALDH1A1ALOX15LMNA
SCHEMBL17177745 0.78 AKR1C2 (0.44) AKR1C2AKR1C1ALDH1A1KMOKDM4E
Biphenyl SCHEMBL2831439 0.77 CES2 (0.56) AKR1C2AKR1C1KMOLMNA
SCHEMBL26352578 0.76 AKR1C2 (0.53) AKR1C2AKR1C1DHODHEGFRKDM4E
SCHEMBL1510357 0.74 AKR1C2 (0.43) AKR1C2AKR1C1DHODHALDH1A1KMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107257803-B Polymyxin antibacterial agents for the treatment of bacterial infections 上海盟科药业股份有限公司 2021-02-05 CN disclosed