SCHEMBL28535555

SCHEMBL28535555

CSc1nc2c(c(OS(=O)(=O)C(F)(F)F)n1)CCCN(Cc1ccccc1)C2

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
C5AR1 P21730 1/20 0.41
GAA P10253 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
ADORA2A P29274 1/20 0.40
KMT2A Q03164 3/20 0.39
CLPP Q16740 6/20 0.37
DRD2 P14416 2/20 0.36
DRD1 P21728 2/20 0.36
DRD4 P21917 2/20 0.36
DRD5 P21918 2/20 0.36
DRD3 P35462 2/20 0.36
MEN1 O00255 1/20 0.36
HTT P42858 1/20 0.36
HRH3 Q9Y5N1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28542677 0.97 KMT2A (0.41) C5AR1GAACYP1A2CYP2C9ADORA2A
SCHEMBL30421340 0.82 TMEM97 (0.41) GAAKMT2A
SCHEMBL30421713 0.82 TMEM97 (0.41) GAAKMT2A
SCHEMBL21315051 0.78 TMEM97 (0.43) GAAKMT2AMEN1
SCHEMBL28503146 0.78 KMT2A (0.31) GAACYP1A2KMT2ADRD2DRD3
SCHEMBL21777116 0.78 KMT2A (0.38) GAACYP1A2KMT2AHTT
SCHEMBL28529445 0.78 GAA (0.42) C5AR1GAACYP1A2CYP2C9ADORA2A
SCHEMBL2341472 0.77 C5AR1 (0.43) C5AR1GAACYP1A2CYP2C9ADORA2A
SCHEMBL26010448 0.76 KMT2A (0.36) GAACYP1A2KMT2AMEN1
SCHEMBL21777078 0.74 CCNA2 (0.37) GAAKMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112538084-B Novel KRAS G12C protein inhibitor and preparation method and application thereof 信达生物制药(苏州)有限公司 2023-06-20 CN disclosed
CN-112538084-A Novel KRAS G12C protein inhibitor and preparation method and application thereof 信达生物制药(苏州)有限公司 2021-03-23 CN disclosed