SCHEMBL28535874

SCHEMBL28535874

O=c1c(I)coc2ccc(-n3cnc(C4CC4)c3)cc12

nearest known ligand 0.56

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 18/20 0.56
CYP17A1 P05093 1/20 0.34
GRM5 P41594 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30095362 1.00 MAP3K5 (0.56) MAP3K5CYP17A1GRM5
SCHEMBL28899163 0.80 MAP3K5 (0.52) MAP3K5
SCHEMBL30095502 0.80 MAP3K5 (0.52) MAP3K5
SCHEMBL28537150 0.79 MAP3K5 (0.52) MAP3K5CYP17A1GRM5
SCHEMBL10222569 0.78 MAP3K5 (0.47) MAP3K5
SCHEMBL23638696 0.73 MAP3K5 (1.00) MAP3K5
SCHEMBL30095507 0.68 IP6K1 (0.55) MAP3K5
SCHEMBL28899189 0.68 IP6K1 (0.55) MAP3K5
SCHEMBL22473968 0.68 MAP3K5 (0.46) MAP3K5
SCHEMBL28899176 0.68 MAP3K5 (0.47) MAP3K5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109456308-B Heterocyclic compounds as ASK inhibitors and their use 南京圣和药业股份有限公司 2022-11-29 CN disclosed
CN-109071498-B Kinase inhibitor and preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2021-03-30 CN disclosed
CN-109456308-A Heterocyclic compound and its application as ASK inhibitor 南京圣和药业股份有限公司 2019-03-12 CN disclosed