SCHEMBL28537150

SCHEMBL28537150

CC1(C)OB(c2coc3ccc(-n4cnc(C5CC5)c4)cc3c2=O)OC1(C)C

nearest known ligand 0.52

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 18/20 0.52
CYP17A1 P05093 1/20 0.33
GRM5 P41594 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28535874 0.79 MAP3K5 (0.56) MAP3K5CYP17A1GRM5
SCHEMBL30095362 0.79 MAP3K5 (0.56) MAP3K5CYP17A1GRM5
SCHEMBL25320169 0.74 LPL (0.38) MAP3K5
SCHEMBL28899163 0.74 MAP3K5 (0.52) MAP3K5
SCHEMBL30095502 0.74 MAP3K5 (0.52) MAP3K5
SCHEMBL25319629 0.73 MAP3K5 (0.41) MAP3K5
SCHEMBL23638696 0.69 MAP3K5 (1.00) MAP3K5
SCHEMBL30095417 0.69 MAP3K5 (1.00) MAP3K5
SCHEMBL25317075 0.66 MAP3K5 (0.39) MAP3K5
SCHEMBL25319660 0.65 MAP3K5 (0.39) MAP3K5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109071498-B Kinase inhibitor and preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2021-03-30 CN disclosed