SCHEMBL28535951

SCHEMBL28535951

C/C(=N\c1ncc(Br)cc1C)C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 5/20 0.41
KDM4E B2RXH2 4/20 0.36
ALDH1A1 P00352 2/20 0.36
CYP1A2 P05177 2/20 0.33
CYP2D6 P10635 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
POLB P06746 1/20 0.33
HCAR2 Q8TDS4 1/20 0.33
RXFP1 Q9HBX9 1/20 0.32
CYP3A4 P08684 1/20 0.32
MAPT P10636 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
ADRA2A P08913 2/20 0.31
ADRA2B P18089 2/20 0.31
ADRA2C P18825 2/20 0.31
TDP1 Q9NUW8 1/20 0.31
RAB9A P51151 3/20 0.31
NPC1 O15118 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25149135 0.81 PLAU (0.43) PLAUALDH1A1MEN1KMT2AADRA2A
SCHEMBL21572709 0.75 PLAU (0.39) PLAUS1PR1S1PR3
SCHEMBL12726178 0.68 KDM4E (0.38) KDM4EALDH1A1CYP1A2MEN1KMT2A
SCHEMBL361806 0.68 KDM4E (0.47) KDM4EALDH1A1POLBHCAR2RXFP1
SCHEMBL25366886 0.66 NPC1 (0.49) KDM4EALDH1A1POLBHCAR2MAPT
SCHEMBL15767643 0.65 AAK1 (0.42) KDM4EALDH1A1CYP1A2CYP2D6MEN1
SCHEMBL760353 0.65 NPC1 (0.48) ALDH1A1MEN1KMT2APOLBMAPT
SCHEMBL12970807 0.65 KDM4E (0.39) KDM4EALDH1A1CYP1A2CYP2D6MEN1
SCHEMBL27751424 0.65 AAK1 (0.42) KDM4EALDH1A1MEN1KMT2APOLB
SCHEMBL29621570 0.63 BACE1 (0.44) PLAUKDM4EALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109053727-B Preparation method of ABT-199 intermediate 山东轩德医药科技有限公司 2021-01-26 CN disclosed