SCHEMBL28537245

SCHEMBL28537245

COO[C@@H]1[C@@H](O)[C@@H](CO)O[C@H]1n1c(Br)nc2c(N)ncnc21

nearest known ligand 0.59

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NADK O95544 2/20 0.59
HSPA5 P11021 2/20 0.58
HSPA8 P11142 2/20 0.58
RXFP1 Q9HBX9 1/20 0.58
HSD17B10 Q99714 1/20 0.52
GAPDH P04406 1/20 0.52
ADORA3 P0DMS8 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30237237 0.92 NADK (0.61) NADKHSPA5HSPA8RXFP1HSD17B10
SCHEMBL5672193 0.92 NADK (0.61) NADKHSPA5HSPA8RXFP1HSD17B10
SCHEMBL1740341 0.92 NADK (0.61) NADKHSPA5HSPA8RXFP1HSD17B10
SCHEMBL28823544 0.86 NADK (0.78) NADKHSPA5HSPA8RXFP1HSD17B10
SCHEMBL12030991 0.85 NADK (0.79) NADKHSPA5HSPA8RXFP1HSD17B10
SCHEMBL13587343 0.85 NADK (0.79) NADKHSPA5HSPA8RXFP1HSD17B10
SCHEMBL1106674 0.85 NADK (0.79) NADKHSPA5HSPA8RXFP1HSD17B10
SCHEMBL440926 0.85 NADK (0.79) NADKHSPA5HSPA8RXFP1HSD17B10
SCHEMBL6671819 0.85 NADK (0.79) NADKHSPA5HSPA8RXFP1HSD17B10
SCHEMBL440925 0.85 NADK (0.79) NADKHSPA5HSPA8RXFP1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112209930-A Istradefylline derivative and preparation method and application thereof 山东新华制药股份有限公司 2021-01-12 CN disclosed