SCHEMBL28537308

SCHEMBL28537308

O=C(O)N1CCc2cc([N+](=O)[O-])c(F)cc2C1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.44
GAA P10253 3/20 0.42
RAB9A P51151 4/20 0.41
CASP3 P42574 1/20 0.40
USP14 P54578 1/20 0.40
UCHL5 Q9Y5K5 1/20 0.40
MAPT P10636 5/20 0.40
ALDH1A1 P00352 3/20 0.39
FAAH O00519 1/20 0.37
MGLL Q99685 1/20 0.37
PDE4B Q07343 1/20 0.37
HTT P42858 1/20 0.37
THRB P10828 1/20 0.37
VDR P11473 1/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
NPC1 O15118 1/20 0.37
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4171865 0.85 ESR1 (0.53) HPGDGAARAB9ACASP3USP14
SCHEMBL29172301 0.84 HPGD (0.45) HPGDGAARAB9AMAPTALDH1A1
SCHEMBL27042944 0.83 HPGD (0.44) HPGDGAARAB9AMAPTALDH1A1
SCHEMBL28711869 0.83 GAA (0.47) HPGDGAARAB9AMAPTALDH1A1
SCHEMBL20214725 0.83 MAPT (0.47) HPGDGAARAB9AMAPTALDH1A1
SCHEMBL4164350 0.82 ESR2 (0.56) HPGDGAARAB9AMAPTALDH1A1
SCHEMBL29741541 0.82 ESR2 (0.56) HPGDGAARAB9AMAPTALDH1A1
SCHEMBL11318782 0.80 MAPT (0.56) RAB9AMAPTALDH1A1HTTTHRB
SCHEMBL29172296 0.80 KDM4E (0.44) HPGDGAARAB9AMAPTALDH1A1
SCHEMBL27042742 0.79 THRA (0.40) HPGDGAARAB9AMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113307772-B Human plasma kallikrein inhibitors 拜奥克里斯特制药公司 2024-06-28 CN disclosed
CN-113307772-A Human plasma kallikrein inhibitors 拜奥克里斯特制药公司 2021-08-27 CN disclosed
CN-106257976-B Human plasma kallikrein inhibitors 拜奥克里斯特制药公司 2021-02-02 CN disclosed