SCHEMBL28537439

SCHEMBL28537439

CC(C)(C)c1c(Oc2nc(-c3nnc(C4CC4)o3)cs2)ccc(OC(N)=O)c1F

nearest known ligand 0.32

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.32
BACE1 P56817 1/20 0.31
BACE2 Q9Y5Z0 1/20 0.31
SMO Q99835 1/20 0.31
TP53 P04637 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23355478 0.81 MAPT (0.34) ATRBACE1BACE2SMOCA1
SCHEMBL21612850 0.74 MAPT (0.33) ATRBACE1BACE2SMO
SCHEMBL28527024 0.74 EIF4E (0.34)
SCHEMBL28527025 0.74
SCHEMBL21612849 0.73 MAPT (0.33) ATRBACE1BACE2
SCHEMBL28526949 0.72 MAP3K14 (0.33)
SCHEMBL28534897 0.72
SCHEMBL24926751 0.69 BRAF (0.40) SMO
SCHEMBL24926748 0.68 BACE1 (0.36) ATRBACE1BACE2CA1CA2
SCHEMBL23355350 0.67 MAPK14 (0.35) SMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112334460-A Biaryl ether type quinazoline derivative 第一三共株式会社 2021-02-05 CN disclosed