SCHEMBL28539764

SCHEMBL28539764

CC(C)(C)OC(=O)N1CCN(c2ncc(C(=O)C(F)(F)F)s2)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 2/20 0.48
HDAC4 P56524 2/20 0.48
HDAC1 Q13547 2/20 0.48
HDAC7 Q8WUI4 2/20 0.48
HDAC2 Q92769 2/20 0.48
HDAC10 Q969S8 2/20 0.48
HDAC11 Q96DB2 2/20 0.48
HDAC8 Q9BY41 2/20 0.48
HDAC6 Q9UBN7 2/20 0.48
HDAC9 Q9UKV0 2/20 0.48
HDAC5 Q9UQL6 2/20 0.48
SCD O00767 3/20 0.46
GPR119 Q8TDV5 6/20 0.44
CKS1B P61024 2/20 0.44
SKP1 P63208 2/20 0.44
SKP2 Q13309 2/20 0.44
HRH3 Q9Y5N1 3/20 0.43
MAPT P10636 2/20 0.41
MEN1 O00255 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2828526 0.90 HDAC3 (0.50) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL2146303 0.86 SCD (0.54) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL16501434 0.86 HDAC3 (0.54) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL13261644 0.85 HRH3 (0.57) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL2575502 0.84 HRH3 (0.58) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL2828808 0.83 HDAC3 (0.48) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL2824232 0.83 CKS1B (0.48) SCDGPR119CKS1BSKP1SKP2
SCHEMBL3155607 0.81 OGA (0.52) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL1199336 0.81 GPR119 (0.49) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL12193543 0.81 HRH3 (0.55) HDAC3HDAC4HDAC1HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105712952-B 2-substituted oxy-5-methylsulfonyl phenyl piperazine amide analogue and preparation method and application thereof 上海翰森生物医药科技有限公司 2021-03-26 CN disclosed