SCHEMBL28539768

SCHEMBL28539768

CCOC(=O)c1cnc(N2CC(c3ccc(C(F)(F)F)cc3)C[C@H]2COCC2CC2)nc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.38
PTGIR P43119 1/20 0.38
ATM Q13315 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
HPGD P15428 1/20 0.36
MAPT P10636 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
CNR2 P34972 1/20 0.36
CCRL2 O00421 1/20 0.36
TRPV1 Q8NER1 1/20 0.35
ACACB O00763 2/20 0.35
POLB P06746 2/20 0.35
FOS P01100 1/20 0.34
JUN P05412 1/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
CNR1 P21554 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28910595 0.90 MAOB (0.38) MAOBATMSMN1; SMN2HPGDMAPT
SCHEMBL28537090 0.88 PTGIR (0.40) PTGIRHRH3ACACBCNR1
SCHEMBL28525724 0.87 MAOB (0.41) MAOBATMSMN1; SMN2HPGDMAPT
SCHEMBL28532378 0.87 MAOB (0.38) MAOBATMSMN1; SMN2HPGDMAPT
SCHEMBL28533221 0.85 MAOB (0.37) MAOBATMSMN1; SMN2HPGDMAPT
SCHEMBL28542465 0.83 MAOB (0.40) MAOBATMSMN1; SMN2HPGDMAPT
SCHEMBL28534572 0.83 MAOB (0.40) MAOBATMSMN1; SMN2HPGDMAPT
SCHEMBL28525878 0.81 KDM4E (0.41) SMN1; SMN2MAPTNPC1RAB9AHRH3
SCHEMBL28526834 0.81 MAOB (0.38) MAOBATMSMN1; SMN2HPGDMAPT
SCHEMBL28526859 0.81 MAOB (0.38) MAOBATMSMN1; SMN2HPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112513021-B ROR gamma antagonist and application thereof in medicines 广东东阳光药业有限公司 2023-06-27 CN disclosed
CN-112513021-A ROR gamma antagonist and application thereof in medicine 广东东阳光药业有限公司 2021-03-16 CN disclosed